tailieunhanh - Pharmaceutical Substances Syntheses, Patents, Applications - Part 182

Pharmaceutical Substances Syntheses, Patents, Applications - Part 182. Reference containing a collection of 2267 active pharmaceutical ingredients, including those launched recently. Listed alphabetically according to their INNs and established a link between INNs, structure, synthesis and production processes, patent and literature situation, medical use, and trade names. For pharmacists and researchers. | Rifampicin R 1811 alternative syntheses DOS 2 537 688 Hoechst appL . JP 54 008 792 Shionogi appl. . JP53 201 155 Suami appl. . Suami T. et al. Carbohydr. Res. CRBRAT 56 415 1977 and literature cited therein. total synthesis Fukami H. et al. Agric. Biol. Chem. ABCHA6 41 1689 1977 . Formulation s vial g 1 g as sulfate Trade Name s D Landamycine Delalande F Ribomycin Delalande I Ibistacin IBI wfm 1977 wfm wfm 1 Vistamycin Meiji 1972 Rifampicin A1C J04AB02 Use antibiotic tuberculosis agent RN 13292-46-1 MF C43H58N4OI2 MW EINECS 236-312-0 LD50 260 mg kg M . 500 mg kg M . 1570 mg kg R . CN 3- 4-methyl-l -piperazinyl imino methyl rifamycin rifomycin B from Streptomyces mediterronei ATCC 13685 rifomycin 0 pyrrolidine 3-pyrrolidinomethyl-rifomycin SV II II 3-formylofamycin SV in 1812 R Rifapentine 1 -omino-4-methyl-piperazine Reference s Maggi N. et al. Chemotherapia CMTRAG 11 285 1966 . US 3 342 810 Lepetit GB-prior. . DAS 1 795 567 Lepetit appl. GB-prior. . alternative synthèses DOS 2 846 321 Holco appl. GB-prior. . fermentative production o rifamycin B DE 1 089 513 Lepetit appl. GB-prior. . Formulation s cps. 150 mg 300 mg drg. 150 mg 300 mg 450 mg 600 mg f. c. tabl. 150 mg 300 mg 450 mg 600 mg syrup 100 mg 5 ml vial 600 mg Trad e Name s D Eremfat Fatol GB Rifa Grünenthal 1970 Rifampicin-Hefa Hefa Pharma Rifater Grünenthal -comb. Rifinah Grünenthal -comb. Rifadin Hoechst 1969 Rifater Hoechst -comb. with isoniazid Rifinah Hoechst -comb. with isoniazid Rimactane Ciba 1969 Rimactane Ciba-Geigy- Fujisawa USA Rifadin Hoechst Marion Roussel 1970 Rifamate Hoechst Marion Roussel 1976 -comb. with F. Rifadine Marion Merrell SA 1969 Rifater Marion Merrell I SA -comb. Rifinah Marion Merrell SA -comb. Rimactan Novartis Pharma J SA 1969 Rimactazid Ciba -comb. with isoniazid Rifadin Lepetit Rifapiam Piam Rifinah Lepetit -comb. with isoniazid Rifadin .